SCHEMBL30786151

SCHEMBL30786151

O=C(NC1CC1)c1ccc(F)cc1Sc1ccc2c(/C=C/c3ccc(CN4CCCC4)cn3)cn(C3CCCCO3)c2c1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 8/20 0.36
KDR P35968 1/20 0.35
KCNH2 Q12809 4/20 0.35
MCHR2 Q969V1 1/20 0.35
CNR1 P21554 4/20 0.34
CNR2 P34972 4/20 0.34
CCR3 P51677 4/20 0.34
ACHE P22303 1/20 0.33
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30786061 0.83 KDR (0.38) MCHR1KDRKCNH2MCHR2CNR1
SCHEMBL31475241 0.82 BDKRB1 (0.32)
SCHEMBL31475185 0.81 KDR (0.34) MCHR1KDRKCNH2
SCHEMBL30786102 0.81 CHEK1 (0.32)
SCHEMBL31576782 0.78 KDR (0.59) MCHR1KDRCCR3
SCHEMBL31475212 0.78 KDR (0.37) KDRCNR1CNR2
SCHEMBL30786153 0.77 KDR (0.36) MCHR1KDRCCR3
SCHEMBL31475215 0.77 KDR (0.37) KDRCNR1CNR2
SCHEMBL31475221 0.76 PRKCQ (0.34)
SCHEMBL31475199 0.76 KDR (0.34) MCHR1KDRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119604488-A Protein tyrosine kinase inhibitor and medical application thereof 苏州必扬医药科技有限公司 2025-03-11 CN disclosed
WO-2024032584-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF 苏州必扬医药科技有限公司 2024-02-15 WO disclosed