SCHEMBL30797273

SCHEMBL30797273

O=C1CCC(N2Cc3cc(N4CCN(c5ccccc5)C4=O)ccc3C2=O)C(=O)N1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 10/20 0.64
CSNK1A1 P48729 1/20 0.58
IKZF1 Q13422 4/20 0.54
IKZF2 Q9UKS7 6/20 0.52
MAP1LC3B Q9GZQ8 1/20 0.50
BRD4 O60885 1/20 0.50
TNF P01375 1/20 0.50
IL1B P01584 1/20 0.50
DDB1 Q16531 1/20 0.50
IKZF3 Q9UKT9 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30797127 0.91 CRBN (0.61) CRBNCSNK1A1IKZF1IKZF2BRD4
SCHEMBL30797106 0.91 CRBN (0.63) CRBNCSNK1A1IKZF1IKZF2
SCHEMBL30797153 0.90 CRBN (0.60) CRBNCSNK1A1IKZF1IKZF2BRD4
SCHEMBL30797297 0.90 CRBN (0.62) CRBNIKZF1IKZF2
SCHEMBL30797195 0.89 CRBN (0.56) CRBNCSNK1A1IKZF1IKZF2MAP1LC3B
SCHEMBL30797266 0.88 CRBN (0.60) CRBNCSNK1A1IKZF1IKZF2DDB1
SCHEMBL30797400 0.88 CRBN (0.60) CRBNCSNK1A1IKZF2
SCHEMBL30797138 0.88 CRBN (0.60) CRBNIKZF1IKZF2
SCHEMBL30797110 0.88 CRBN (0.60) CRBNCSNK1A1IKZF2DDB1
SCHEMBL30797338 0.88 CRBN (0.64) CRBNCSNK1A1IKZF1IKZF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023244817-A1 SUBSTITUTED PIPERIDINES AS CK1A DEGRADERS MONTE ROSA THERAPEUTICS, INC. (US) 2023-12-21 WO disclosed