SCHEMBL30801290

SCHEMBL30801290

O=C1c2ccc(N3CCC(C4OCCO4)CC3)cc2CN1C1CCCNC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
HTR2B P41595 13/20 0.38
HTR2C P28335 13/20 0.38
HTR2A P28223 12/20 0.38
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CRBN Q96SW2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29966331 0.85 PARP1 (0.46) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL29966514 0.85 PARP1 (0.46) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL26625271 0.85 PARP1 (0.46) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL30702597 0.82 PARP1 (0.40) PARP1HTR2BHTR2CHTR2AALDH1A1
SCHEMBL30002807 0.81 PARP1 (0.44) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL30595369 0.80 PARP1 (0.42) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL32664871 0.80 PARP1 (0.41) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL30635212 0.80 HTR2C (0.41) PARP1HTR2BHTR2CHTR2AMEN1
SCHEMBL30635240 0.80 HTR2C (0.41) PARP1HTR2BHTR2CHTR2AMEN1
SCHEMBL30351677 0.79 PARP1 (0.43) PARP1HTR2BHTR2CHTR2AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117693502-A Compounds for inhibiting or degrading ITK, compositions comprising the same, methods of making the same, and methods of using the same 纽力克斯治疗公司 2024-03-12 CN disclosed