SCHEMBL30811237

SCHEMBL30811237

CCCCc1ccc(NCc2ccc(-c3nc4c(C(N)=O)cccc4[nH]3)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.68
HDAC3 O15379 1/20 0.64
HDAC1 Q13547 1/20 0.64
HDAC2 Q92769 1/20 0.64
PARP2 Q9UGN5 1/20 0.64
DHODH Q02127 2/20 0.59
AURKA O14965 1/20 0.55
AURKB Q96GD4 1/20 0.55
PLA2G2A P14555 1/20 0.54
ALOX15 P16050 1/20 0.54
PTGS2 P35354 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29180033 1.00 PARP1 (0.68) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL30811253 0.90 PARP1 (0.73) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL29180031 0.90 PARP1 (0.73) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL29179987 0.87 PARP1 (0.74) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL29179990 0.85 PARP1 (0.77) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL30811239 0.85 PARP1 (0.77) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL29180021 0.84 PARP1 (0.73) PARP1PARP2DHODHAURKAAURKB
SCHEMBL30811254 0.83 PARP1 (0.72) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL29180003 0.83 PARP1 (0.72) PARP1HDAC3HDAC1HDAC2PARP2
SCHEMBL30811248 0.82 PARP1 (0.70) PARP1HDAC3HDAC1HDAC2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117624054-A PARP inhibitor 2-substituted benzimidazole compound, and preparation method and application thereof 广西大学 2024-03-01 CN disclosed