SCHEMBL30816005

SCHEMBL30816005

O=C1Nc2cc(Br)cnc2N2CCN(C(=O)OCc3ccccc3)CC12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GRIN2B Q13224 4/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
USP30 Q70CQ3 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
F13A1 P00488 1/20 0.38
TGM2 P21980 1/20 0.38
TGM1 P22735 1/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPK1 P28482 2/20 0.38
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102338 1.00 SMN1; SMN2 (0.40) SMN1; SMN2NPC1RAB9AGRIN2BNR1H2
SCHEMBL29274281 0.87 CBLB (0.49) SMN1; SMN2NPC1RAB9AGRIN2BNR1H2
SCHEMBL11487880 0.85 GRIN2B (0.45) SMN1; SMN2NPC1RAB9AGRIN2BCYP2C19
SCHEMBL5129484 0.84 SMN1; SMN2 (0.42) SMN1; SMN2NPC1RAB9AUSP30CYP2C19
SCHEMBL30816015 0.83 GRIN2B (0.41) SMN1; SMN2NPC1RAB9AGRIN2BNR1H2
SCHEMBL23102342 0.83 GRIN2B (0.41) SMN1; SMN2NPC1RAB9AGRIN2BNR1H2
SCHEMBL29170650 0.82 KDM4E (0.46) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL11477857 0.80 SMN1; SMN2 (0.42) SMN1; SMN2NPC1RAB9AGRIN2BNR1H2
SCHEMBL23102322 0.80 KDM4E (0.43) MEN1KMT2AHDAC6KDM4EALDH1A1
SCHEMBL23102324 0.80 KDM4E (0.43) MEN1KMT2AHDAC6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114096533-B Tri-ring compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-03-08 CN disclosed