SCHEMBL30833400

SCHEMBL30833400

Cc1cc(NC(=O)N2CCC(C(C)(F)S(=O)(=O)c3cccc(F)c3)CC2)cnn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
NPC1 O15118 1/20 0.44
CYP3A4 P08684 2/20 0.43
NR1I2 O75469 1/20 0.43
CACNA1B Q00975 1/20 0.43
KMT2A Q03164 1/20 0.42
ABCC9 O60706 1/20 0.41
ABCC8 Q09428 1/20 0.41
KCNJ11 Q14654 1/20 0.41
KCNJ8 Q15842 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
HPGDS O60760 1/20 0.40
CYP2C9 P11712 5/20 0.40
USP2 O75604 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HIF1A Q16665 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17942430 1.00 TSHR (0.47) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL17949199 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL30833428 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL29529870 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL29529953 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL17949166 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL17949198 0.88 TSHR (0.48) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL29529596 0.88 TSHR (0.47) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL17949479 0.88 TSHR (0.47) TSHRNPC1CYP3A4NR1I2CACNA1B
SCHEMBL17949486 0.87 TSHR (0.49) TSHRNPC1CYP3A4NR1I2CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118164961-A 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-06-11 CN disclosed
CN-111393414-B 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-05-07 CN disclosed