SCHEMBL30834547

SCHEMBL30834547

COc1cc(C2Cc3ncnc(N4CCNCC4)c3CC2C)c2ccccc2c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2C19 P33261 3/20 0.42
CLK4 Q9HAZ1 3/20 0.42
USP2 O75604 2/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
HTR2C P28335 2/20 0.38
TOP1 P11387 3/20 0.37
KRAS P01116 1/20 0.37
HTR6 P50406 2/20 0.36
ADRB1 P08588 1/20 0.36
PRMT5 O14744 1/20 0.36
NCF1 P14598 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21733840 1.00 CYP1A2 (0.42) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL30834507 0.87 KRAS (0.42) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL21733676 0.87 KRAS (0.42) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL21722152 0.84 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL30834556 0.84 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL21722298 0.80 TLR7 (0.41) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL21722193 0.76 KRAS (0.54) KRAS
SCHEMBL29697525 0.76 KRAS (0.53) CYP1A2CYP3A4CYP2C19CLK4USP2
SCHEMBL21722230 0.75 SRC (0.38) ALDH1A1TP53
SCHEMBL30834559 0.75 SRC (0.38) ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112119075-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-12 CN disclosed