SCHEMBL30834553

SCHEMBL30834553

CC1Cc2c(ncnc2N2CCNCC2)CC1c1nc(N)ccc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.38
EPHX2 P34913 1/20 0.38
CYP1A2 P05177 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KRAS P01116 4/20 0.36
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
CYP2C19 P33261 1/20 0.35
RPS6KB1 P23443 5/20 0.35
AKT1 P31749 3/20 0.35
ADRB2 P07550 1/20 0.34
NCF1 P14598 1/20 0.34
CNR2 P34972 1/20 0.34
CYP2C9 P11712 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24855323 0.84 EPHX2 (0.34) HRH4EPHX2CYP1A2KDM4EALDH1A1
SCHEMBL29191281 0.83 KRAS (0.45) HRH4CYP1A2ALDH1A1KRASCYP2C19
SCHEMBL21733596 0.83 KRAS (0.53) KRAS
SCHEMBL21734100 0.83 KRAS (0.53) KRAS
SCHEMBL21733900 0.83 KRAS (0.53) KRAS
SCHEMBL30178116 0.83 KRAS (0.53) KRAS
SCHEMBL21722245 0.83 KRAS (0.53) KRAS
SCHEMBL21722148 0.83 KRAS (0.53) KRAS
SCHEMBL29191268 0.82 EPHX2 (0.38) HRH4EPHX2CYP1A2KRASCYP2C19
SCHEMBL30834529 0.82 EPHX2 (0.38) HRH4EPHX2CYP1A2KRASCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112119075-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-12 CN disclosed