SCHEMBL30851263

SCHEMBL30851263

COc1ncc(CCN)cc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.45
HTR2C P28335 3/20 0.45
HTR2B P41595 2/20 0.38
AURKA O14965 1/20 0.37
KDR P35968 1/20 0.37
AURKB Q96GD4 1/20 0.37
MAOB P27338 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ATM Q13315 1/20 0.37
TAAR1 Q96RJ0 6/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24968405 1.00 HTR2A (0.45) HTR2AHTR2CHTR2BAURKAKDR
SCHEMBL24968228 0.84 AURKA (0.37) HTR2AHTR2CAURKAKDRAURKB
SCHEMBL30851115 0.84 AURKA (0.37) HTR2AHTR2CAURKAKDRAURKB
SCHEMBL21031170 0.82 AURKA (0.40) HTR2AHTR2CAURKAKDRAURKB
SCHEMBL24968232 0.82 ATM (0.40) AURKAKDRAURKBATMTAAR1
SCHEMBL30851096 0.82 ATM (0.40) AURKAKDRAURKBATMTAAR1
SCHEMBL932942 0.81 AURKA (0.39) AURKAKDRAURKBPIK3R1PIK3CA
SCHEMBL29208803 0.81 AURKA (0.39) AURKAKDRAURKBPIK3R1PIK3CA
SCHEMBL27233788 0.81 AURKA (0.39) HTR2AHTR2CAURKAKDRAURKB
SCHEMBL29165939 0.79 PIK3R1 (0.36) AURKAKDRAURKBKDM4EPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117642393-A Novel PARP7 inhibitor and application thereof 上海齐鲁制药研究中心有限公司 2024-03-01 CN disclosed