SCHEMBL30860

SCHEMBL30860

O=C1c2cc(Br)ccc2CC12CCC1=C(CCC=C1)CC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PARP1 P09874 1/20 0.33
PARP10 Q53GL7 1/20 0.33
TGM2 P21980 1/20 0.33
CES1 P23141 1/20 0.33
METAP1 P53582 1/20 0.31
TDP2 O95551 1/20 0.31
HSP90AA1 P07900 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
KDM1A O60341 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7879908 0.86 TDP1 (0.35) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL30642 0.86 TDP1 (0.35) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL30482 0.79 TDP1 (0.45) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL1465537 0.79 TDP1 (0.41) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL9948162 0.78 TDP1 (0.46) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL7887048 0.77 TDP1 (0.33) TDP1L3MBTL1PARP1PARP10
SCHEMBL30859 0.77 TDP1 (0.41) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL30785 0.76 TDP1 (0.54) TDP1L3MBTL1PARP1PARP10CA1
SCHEMBL9948561 0.75 TDP1 (0.44) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL28187 0.75 HDAC3 (0.35) TDP1L3MBTL1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406240-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2012-01-18 EP disclosed
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed