SCHEMBL30872161

SCHEMBL30872161

Cc1cc(C)nc(-n2cc3c(c2)CN(C(=O)c2c(-c4ccccn4)cn4ccccc24)C3)n1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.48
HCRTR2 O43614 19/20 0.48
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40
BAZ2B Q9UIF8 1/20 0.40
BAZ2A Q9UIF9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30872176 0.87 KDM4E (0.47) HCRTR1HCRTR2
SCHEMBL30872171 0.86 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL30872186 0.85 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL30872184 0.84 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL30872174 0.83 HCRTR1 (0.35) HCRTR1HCRTR2
SCHEMBL31351492 0.83 HCRTR1 (0.68) HCRTR1HCRTR2
SCHEMBL30872180 0.83 HCRTR1 (0.43) HCRTR1HCRTR2BRD4BRD2BRD3
SCHEMBL30872177 0.75 HCRTR1 (0.65) HCRTR1HCRTR2
SCHEMBL30872162 0.73 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL30872157 0.72 HCRTR2 (0.70) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024109672-A1 DISUBSTITUTED OCTAHYDROPYRROLO[3,4-C]PYRROLE METHYL KETONE DERIVATIVE AND APPLICATION THEREOF 江苏恩华药业股份有限公司 2024-05-30 WO disclosed