SCHEMBL30877064

SCHEMBL30877064

NC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)cc3C(F)(F)F)c(F)c2)cc[n+]1[O-]

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 9/20 0.42
KDR P35968 8/20 0.42
MAPK14 Q16539 2/20 0.42
RIPK2 O43353 1/20 0.42
ABCB11 O95342 1/20 0.42
ABL1 P00519 1/20 0.42
RAF1 P04049 1/20 0.42
NR3C1 P04150 1/20 0.42
RET P07949 1/20 0.42
HTR1A P08908 1/20 0.42
PDGFRB P09619 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
KIT P10721 1/20 0.42
CHRM1 P11229 1/20 0.42
BCR P11274 1/20 0.42
FGFR1 P11362 1/20 0.42
RARG P13631 1/20 0.42
PDGFRA P16234 1/20 0.42
FLT1 P17948 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15114775 0.86 KDR (0.58) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL29746649 0.86 KDR (0.58) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL29523346 0.82 KDR (0.59) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL15114776 0.78 KDR (0.68) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL29746661 0.78 KDR (0.68) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL14714846 0.77 KDR (0.62) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL548163 0.76 RAF1 (0.64) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL5502095 0.74 KDR (0.61) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL548196 0.72 RAF1 (0.55) BRAFKDRMAPK14RIPK2ABCB11
SCHEMBL4255951 0.69 KDR (0.67) BRAFKDRMAPK14RIPK2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11951166-B2 Combination of regorafenib and PD-1/PD-L1(2) inhibitors for treating cancer BAYER AKTIENGESELLSCHAFT (DE) 2024-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11951166-B2 Combination of regorafenib and PD-1/PD-L1(2) inhibitors for treating cancer PDCD1, CD274, PDCD1LG2 BRAF 9/4885KDR 1071/4885MAPK14 1406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.