SCHEMBL30912484

SCHEMBL30912484

CN1C(=O)CCC1c1ccc(N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
THRB P10828 2/20 0.54
TSHR P16473 2/20 0.54
CYP3A4 P08684 1/20 0.54
THPO P40225 1/20 0.54
MEN1 O00255 1/20 0.54
MAPK1 P28482 1/20 0.54
KMT2A Q03164 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
CYP19A1 P11511 7/20 0.47
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
LMNA P02545 1/20 0.40
APEX1 P27695 1/20 0.40
PMP22 Q01453 1/20 0.40
NFKB1 P19838 1/20 0.40
CYP2C19 P33261 1/20 0.40
SRD5A1 P18405 5/20 0.38
SRD5A2 P31213 1/20 0.37
CYP11B1 P15538 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30912593 1.00 KDM4E (0.54) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL30912576 1.00 KDM4E (0.54) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL13521128 0.82 CYP3A4 (0.54) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL22781363 0.82 SRD5A1 (0.57) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL3140704 0.82 CYP3A4 (0.54) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL13225803 0.81 KDM4E (0.66) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL11708369 0.81 KDM4E (0.66) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL5309109 0.76 CYP19A1 (0.41) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL30912493 0.76 KDM4E (0.48) KDM4ETHRBTSHRCYP3A4THPO
SCHEMBL9414375 0.75 TSHR (0.50) KDM4ETHRBTSHRCYP3A4THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4619406-A1 TRICYCLIC COMPOUNDS Schrödinger, Inc. (US) 2025-09-24 EP disclosed
WO-2024107393-A1 TRICYCLIC COMPOUNDS SCHRÖDINGER, INC. (US) 2024-05-23 WO disclosed