SCHEMBL30917869

SCHEMBL30917869

Cc1nc2ccc(-c3nc(Nc4ccc(CN5CCN(C(C)C)CC5)cn4)ncc3F)cc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 12/20 1.00
CDK6 Q00534 7/20 0.78
CCND1 P24385 4/20 0.69
CDK4 P11802 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29230288 1.00 DYRK2 (1.00) DYRK2CDK6CCND1CDK4
SCHEMBL32677350 0.91 DYRK2 (1.00) DYRK2CDK6CCND1CDK4
SCHEMBL26447899 0.91 DYRK2 (1.00) DYRK2CDK6CCND1CDK4
SCHEMBL26448508 0.91 DYRK2 (0.87) DYRK2CDK6CCND1CDK4
SCHEMBL30569702 0.90 DYRK2 (0.81) DYRK2CDK6CCND1CDK4
SCHEMBL26447961 0.90 DYRK2 (0.81) DYRK2CDK6CCND1CDK4
SCHEMBL26447911 0.89 DYRK2 (0.98) DYRK2CDK6CCND1
SCHEMBL26447989 0.88 DYRK2 (0.79) DYRK2CDK6CCND1CDK4
Hydrochloric Acid SCHEMBL29754498 0.88 DYRK2 (1.00) DYRK2CDK6CCND1
Hydrochloric Acid SCHEMBL26679973 0.88 DYRK2 (1.00) DYRK2CDK6CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4631941-A1 BENZOTHIAZOLE PYRIMIDINEAMINE DYRK2 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF Jiangsu Tasly Diyi Pharmaceutical Co., Ltd. (CN) 2025-10-15 EP disclosed
CN-118146213-B Benzothiazole pyrimidine amine DYRK2 inhibitor and preparation method and application thereof 江苏天士力帝益药业有限公司 2024-11-26 CN disclosed
CN-118146213-A Benzothiazole pyrimidine amine DYRK2 inhibitor and preparation method and application thereof 江苏天士力帝益药业有限公司 2024-06-07 CN disclosed