SCHEMBL30946641

SCHEMBL30946641

COc1cnc2c(O)ncnc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.41
MAPK7 Q13164 1/20 0.38
BACE1 P56817 6/20 0.35
CTSD P07339 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
HPGDS O60760 2/20 0.34
BACE2 Q9Y5Z0 3/20 0.34
MAP4K4 O95819 1/20 0.33
ALDH1A1 P00352 1/20 0.33
F2 P00734 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
PDE10A Q9Y233 1/20 0.33
MAPT P10636 1/20 0.33
GRM1 Q13255 1/20 0.33
PDE6D O43924 1/20 0.32
PDE6A P16499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21219055 1.00 EGFR (0.41) EGFRMAPK7BACE1CTSDCYP1A1
SCHEMBL15900276 0.79 KMT2A (0.43) EGFRMAPK7BACE1CTSDCYP1A1
SCHEMBL16485382 0.78 EGFR (0.38) EGFRMAPK7BACE1CTSDCYP1A1
SCHEMBL20568790 0.76 CCR1 (0.42)
SCHEMBL23170997 0.74 TLR8 (0.43) EGFR
SCHEMBL22872946 0.72
SCHEMBL21219052 0.72 GRIN2D (0.33) BACE1CTSDBACE2
SCHEMBL4978434 0.72 DYRK1A (0.37) BACE1BACE2ALDH1A1MAPT
SCHEMBL30946648 0.72 GRIN2D (0.33) BACE1CTSDBACE2
SCHEMBL4295596 0.71 ESR1 (0.47) EGFRCYP1A1CYP1B1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112312909-B Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-07-02 CN disclosed