SCHEMBL30948587

SCHEMBL30948587

CP(C)c1c(Nc2nc(Nc3ccc(F)c([N+](=O)[O-])c3)ncc2Br)ccc2nccnc12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 8/20 0.41
EGFR P00533 4/20 0.40
ABCG2 Q9UNQ0 3/20 0.37
ZAP70 P43403 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.36
PTK2B Q14289 1/20 0.36
CDK2 P24941 1/20 0.35
KDR P35968 1/20 0.35
GSK3B P49841 1/20 0.35
STK17A Q9UEE5 1/20 0.35
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29253659 1.00 CDK1 (0.41) CDK1EGFRABCG2ZAP70MEN1
SCHEMBL28650588 0.90 BRD4 (0.40) ABCG2MEN1CYP1A2CYP3A4MAPT
SCHEMBL30948628 0.90 BRD4 (0.40) ABCG2MEN1CYP1A2CYP3A4MAPT
SCHEMBL28650090 0.86 EGFR (0.48) EGFR
SCHEMBL30948581 0.81 EGFR (0.40) EGFR
SCHEMBL30948586 0.79 EGFR (0.44) EGFR
SCHEMBL30948609 0.79 ABCG2 (0.41) ABCG2ZAP70CDK2STK17A
SCHEMBL30626557 0.78 EGFR (0.45) EGFRZAP70MEN1MAPTKMT2A
SCHEMBL28531353 0.78 EGFR (0.45) EGFRZAP70MEN1MAPTKMT2A
SCHEMBL25002512 0.77 IGF1R (0.39) CDK1EGFRZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed