SCHEMBL30957500

SCHEMBL30957500

COc1cnc(Cl)nc1-c1c[nH]c2c(C)cccc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.47
CCNT1 O60563 3/20 0.44
CCNK O75909 3/20 0.44
CCNE1 P24864 3/20 0.44
CDK2 P24941 3/20 0.44
CDK9 P50750 3/20 0.44
CDK12 Q9NYV4 3/20 0.44
RPS6KA5 O75582 1/20 0.43
DYRK1A Q13627 2/20 0.43
NFATC1 O95644 1/20 0.43
GSK3B P49841 1/20 0.43
NR4A2 P43354 1/20 0.41
ATP4A P20648 1/20 0.40
ATP4B P51164 1/20 0.40
CDK7 P50613 2/20 0.40
CCNH P51946 2/20 0.40
MNAT1 P51948 2/20 0.40
CLK1 P49759 1/20 0.39
JAK1 P23458 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24900366 1.00 AR (0.47) ARCCNT1CCNKCCNE1CDK2
SCHEMBL30957550 0.90 DYRK1A (0.53) ARRPS6KA5DYRK1ANFATC1GSK3B
SCHEMBL24900358 0.90 DYRK1A (0.53) ARRPS6KA5DYRK1ANFATC1GSK3B
SCHEMBL30957556 0.87 CCNT1 (0.43) ARCCNT1CCNKCCNE1CDK2
SCHEMBL24900454 0.87 CCNT1 (0.43) ARCCNT1CCNKCCNE1CDK2
SCHEMBL24900582 0.85 RPS6KA5 (0.60) ARCCNT1CCNKCCNE1CDK2
SCHEMBL30957639 0.82 CCNT1 (0.55) ARCCNT1CCNKCCNE1CDK2
SCHEMBL24900677 0.82 CCNT1 (0.55) ARCCNT1CCNKCCNE1CDK2
SCHEMBL24900727 0.81 RPS6KA5 (0.56) ARCCNT1CCNKCCNE1CDK2
SCHEMBL17542563 0.81 CDK7 (0.54) RPS6KA5CDK7CCNHMNAT1CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118159533-A Heterocyclic compounds and their use 艾森医药有限公司 2024-06-07 CN disclosed