SCHEMBL30980951

SCHEMBL30980951

Nc1cc(Br)ccc1N[C@H]1CCOC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 6/20 0.41
BACE1 P56817 2/20 0.37
BACE2 Q9Y5Z0 2/20 0.37
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE1C Q14123 1/20 0.34
ALOX15 P16050 2/20 0.33
CD38 P28907 1/20 0.33
BRD4 O60885 3/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23177187 1.00 AAK1 (0.41) AAK1BACE1BACE2KDM1AMAOA
SCHEMBL28536662 1.00 AAK1 (0.41) AAK1BACE1BACE2KDM1AMAOA
SCHEMBL23177336 1.00 AAK1 (0.41) AAK1BACE1BACE2KDM1AMAOA
SCHEMBL29791971 0.91 AAK1 (0.44) AAK1KDM1AMAOAMAOBKDM4E
SCHEMBL2687892 0.91 AAK1 (0.44) AAK1KDM1AMAOAMAOBKDM4E
SCHEMBL28627251 0.87 AAK1 (0.41) AAK1KDM4EGAAMAPTALOX15
SCHEMBL29502212 0.82 AAK1 (0.48) AAK1KDM4EGAAMAPTALOX15
SCHEMBL459719 0.82 AAK1 (0.48) AAK1KDM4EGAAMAPTALOX15
SCHEMBL27007895 0.80 AAK1 (0.43) AAK1KDM1AMAOAMAOBMAPT
SCHEMBL12820435 0.79 HSP90AA1 (0.48) AAK1BACE1BACE2HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574189-B EP300/CBP inhibitor 海创药业股份有限公司 2024-05-31 CN disclosed