SCHEMBL30990907

SCHEMBL30990907

COc1cc2c(=O)n(CCN3CCN(C)CC3)c3c4cc5c(cc4ccc3c2cc1OC)OCO5

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 17/20 0.69
ABCC1 P33527 1/20 0.46
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21630106 1.00 TDP1 (0.69) TDP1ABCC1KDM4EALDH1A1MAPK1
SCHEMBL30990879 0.94 TDP1 (0.67) TDP1ABCC1MAPK1
SCHEMBL21630147 0.94 TDP1 (0.67) TDP1ABCC1MAPK1
SCHEMBL21630163 0.93 TDP1 (0.71) TDP1ABCC1KDM4EMAPK1
SCHEMBL30990883 0.93 TDP1 (0.71) TDP1ABCC1KDM4EMAPK1
SCHEMBL21630157 0.92 TDP1 (0.69) TDP1ABCC1MAPK1
SCHEMBL30990888 0.92 TDP1 (0.69) TDP1ABCC1MAPK1
SCHEMBL21630127 0.92 TDP1 (0.69) TDP1ABCC1KDM4EMAPK1
SCHEMBL30990898 0.92 TDP1 (0.69) TDP1ABCC1KDM4EMAPK1
SCHEMBL21630174 0.88 TDP1 (0.66) TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114555189-B Zanthoxylum nitidum base derivatives as inhibitors of topoisomerase IB (TOP 1) and/or tyrosyl-DNA phosphodiesterase 1 (TDP 1) 美国政府健康及人类服务部 2024-08-02 CN disclosed