SCHEMBL3108263

SCHEMBL3108263

CCOC(=O)Cn1nnc(-c2cc(OC3CCC(Oc4cc(Cl)ccc4Br)CC3)no2)n1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.53
SCD5 Q86SK9 2/20 0.46
ALDH1A1 P00352 3/20 0.40
MAPK1 P28482 1/20 0.40
MAPT P10636 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
XPO1 O14980 1/20 0.39
HTT P42858 3/20 0.37
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KMT2A Q03164 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3321553 0.90 SCD (0.64) SCDSCD5
SCHEMBL13332472 0.87 SCD (0.61) SCDSCD5ALDH1A1MAPK1MAPT
SCHEMBL13361544 0.84 SCD (0.48) SCDSCD5
SCHEMBL3261795 0.83 SCD (0.46) SCDSCD5ALDH1A1MAPK1HPGD
SCHEMBL3320133 0.78 SCD (0.64) SCDSCD5ALDH1A1POLBLMNA
SCHEMBL3320435 0.77 SCD (0.74) SCDSCD5
SCHEMBL3328862 0.76 SCD (0.63) SCDSCD5
SCHEMBL3323795 0.75 SCD (0.60) SCDSCD5ALDH1A1XPO1POLB
SCHEMBL13332435 0.73 SCD (0.53) SCDSCD5ALDH1A1MAPK1MAPT
SCHEMBL13361526 0.72 SCD (0.48) SCDSCD5ALDH1A1XPO1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148878-A1 NOVEL HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Frosst Canada Ltd. (CA) 2010-02-03 EP disclosed
WO-2008128335-A1 NOVEL HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2008-10-30 WO disclosed