SCHEMBL31089002

SCHEMBL31089002

CCOC(=O)C[C@H](N[S@+]([O-])C(C)(C)C)c1cc(Br)ccc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
ALOX5 P09917 3/20 0.35
KAT6A Q92794 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 2/20 0.34
BACE1 P56817 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
AAK1 Q2M2I8 1/20 0.32
FPR2 P25090 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24036886 0.90 MEN1 (0.34) KAT6AALDH1A1BACE1HPGDKMT2A
SCHEMBL25753621 0.90 MEN1 (0.34) KAT6AALDH1A1BACE1HPGDKMT2A
SCHEMBL28957391 0.88 BACE1 (0.34) NPSR1BACE1
SCHEMBL29725911 0.88 BACE1 (0.34) NPSR1BACE1
SCHEMBL31089151 0.88 TSHR (0.39) NPSR1ADORA3SMN1; SMN2ALDH1A1MAPT
SCHEMBL29725964 0.86 BACE1 (0.34) NPSR1BACE1
SCHEMBL31088888 0.86 BACE1 (0.33) BACE1
SCHEMBL25819422 0.86 BACE1 (0.34) NPSR1BACE1
SCHEMBL23259944 0.86 BACE1 (0.34) NPSR1BACE1
SCHEMBL30972783 0.85 BACE1 (0.35) NPSR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175907-A1 MACROCYCLIC ALPHA4BETA7 INTEGRIN INHIBITORS C4X DISCOVERY LIMITED (GB) 2024-08-29 WO disclosed