SCHEMBL31249971

SCHEMBL31249971

CCOC(=O)c1cncc(Br)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46
MAPT P10636 3/20 0.44
ALDH1A1 P00352 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
POLB P06746 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
PKM P14618 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HTT P42858 1/20 0.41
GAA P10253 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8884008 1.00 CYP1A2 (0.51) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL4338257 0.82 CYP1A2 (0.55) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL164287 0.81 CYP1A2 (0.53) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL17440722 0.80 MRGPRX4 (0.43) CYP1A2MAPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL14825220 0.80 CYP1A2 (0.49) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL6202564 0.80 CYP1A2 (0.53) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL3697022 0.79 CYP1A2 (0.51) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL12228820 0.79 CYP1A2 (0.51) CYP1A2CYP2C19CYP2C9MAPTALDH1A1
SCHEMBL29911292 0.76 CYP1A2 (0.77) CYP1A2MAPTALDH1A1NPC1RAB9A
SCHEMBL198054 0.76 CYP1A2 (0.77) CYP1A2MAPTALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118684631-A External nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP 1) inhibitors, compositions and uses thereof 中国科学院上海药物研究所 2024-09-24 CN disclosed