SCHEMBL31267397

SCHEMBL31267397

CN(C)C(=O)c1cc2cnc(Cl)nc2n1-c1ccc2c(c1)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
NR1H2 P55055 2/20 0.43
CDK2 P24941 2/20 0.41
MAPT P10636 2/20 0.39
AURKA O14965 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CDK4 P11802 4/20 0.37
QRFPR Q96P65 2/20 0.37
HDAC1 Q13547 1/20 0.36
IGF1R P08069 1/20 0.36
NR1H3 Q13133 1/20 0.35
MAP3K5 Q99683 1/20 0.35
CDK1 P06493 1/20 0.35
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
PTK2 Q05397 1/20 0.35
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30643145 1.00 ESR2 (0.50) ESR2NR1H2CDK2MAPTAURKA
SCHEMBL2303422 0.74 CDK4 (0.51) CDK2AURKACDK4CDK1
SCHEMBL26637834 0.73 CDK4 (0.41) CDK2CDK4CDK1
SCHEMBL30368378 0.73 ESR2 (0.67) ESR2NR1H2MAPTHDAC1
SCHEMBL30301704 0.73 ESR2 (0.67) ESR2NR1H2MAPTHDAC1
SCHEMBL2304507 0.71 CDK4 (0.47) CDK2CDK4HDAC1CDK1
SCHEMBL26638064 0.71 CDK4 (0.41) CDK2CDK4CDK1
SCHEMBL12518355 0.70 ESR2 (0.55) ESR2NR1H2CDK2MAPTIGF1R
SCHEMBL31621670 0.70 ESR2 (0.78) ESR2NR1H2LMNATP53HDAC1
SCHEMBL19684692 0.70 ESR2 (0.78) ESR2NR1H2LMNATP53HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119156389-A Heterocyclic compounds, compositions thereof and methods of treatment thereof 百济神州有限公司 2024-12-17 CN disclosed