SCHEMBL31276014

SCHEMBL31276014

COC(=O)c1ccc2c(c1)CCN(C(C)=O)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 6/20 0.56
HDAC8 Q9BY41 2/20 0.56
NOTUM Q6P988 1/20 0.56
ACACB O00763 1/20 0.52
PRMT5 O14744 2/20 0.50
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
MAPK1 P28482 1/20 0.48
NAMPT P43490 3/20 0.47
EP300 Q09472 2/20 0.47
CREBBP Q92793 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
BRD4 O60885 1/20 0.47
TMPRSS2 O15393 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12682930 1.00 HDAC6 (0.56) HDAC6HDAC8NOTUMACACBPRMT5
SCHEMBL17560214 0.94 NOTUM (0.56) HDAC6HDAC8NOTUMACACBPRMT5
SCHEMBL1027755 0.89 HDAC6 (0.56) HDAC6HDAC8ACACBESR1ESR2
SCHEMBL1263724 0.85 HDAC6 (0.53) HDAC6HDAC8ACACBESR1ESR2
SCHEMBL8283285 0.85 ESR2 (0.70) HDAC6HDAC8ACACBESR1ESR2
SCHEMBL1027560 0.84 HDAC6 (0.73) HDAC6HDAC8NOTUMPRMT5HDAC3
SCHEMBL20178664 0.84 HDAC6 (0.51) HDAC6HDAC8ACACBESR1ESR2
SCHEMBL10120405 0.84 HDAC6 (0.52) HDAC6HDAC8ACACBESR1ESR2
SCHEMBL17560164 0.84 NOTUM (0.61) HDAC6HDAC8NOTUMPRMT5ESR1
SCHEMBL30810841 0.83 HDAC6 (0.51) HDAC6HDAC8ACACBESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119173512-A Small molecule inhibitors of ubiquitin-specific protease 1 (USP 1) and uses thereof 英矽智能科技知识产权有限公司 2024-12-20 CN disclosed