SCHEMBL31310189

SCHEMBL31310189

CC(C)(O)c1ccn2nc(Br)nc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.36
CYP11B2 P19099 1/20 0.33
PDE10A Q9Y233 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PIK3CD O00329 1/20 0.30
PAK4 O96013 1/20 0.30
JAK1 P23458 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
CSNK1A1 P48729 1/20 0.30
PIK3CG P48736 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
PIP4K2C Q8TBX8 1/20 0.30
CSNK1G1 Q9HCP0 1/20 0.30
NR4A2 P43354 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12077911 0.80 PDE10A (0.43) AHRPDE10AKDM4EALDH1A1
SCHEMBL20605163 0.74 KDM4E (0.41) AHRCYP11B2PDE10AKDM4EALDH1A1
SCHEMBL15539271 0.74 AHR (0.41) AHRPDE10AKDM4EALDH1A1MAPK1
SCHEMBL31456654 0.74 AHR (0.41) AHR
SCHEMBL31264174 0.72 AURKA (0.43) AHRALDH1A1MAPK1L3MBTL1
SCHEMBL31310205 0.71 AHR (0.36) AHRNR4A2
SCHEMBL20986019 0.71 AHR (0.50) AHR
SCHEMBL30842034 0.70 CYP11B1 (0.46) AHRCYP11B2PIK3CDPIK3CAPIK3CG
SCHEMBL9105398 0.70 AHR (0.41) AHRCYP11B2KDM4EALDH1A1PIK3CD
SCHEMBL31456625 0.70 AHR (0.38) AHRCYP11B2KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119264042-A Cyclopentane derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2025-01-07 CN disclosed