SCHEMBL3131699

SCHEMBL3131699

Cc1oc(CCC(N)=O)nc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.43
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
KLF5 Q13887 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.35
RXRA P19793 7/20 0.33
IKBKB O14920 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
BMP1 P13497 1/20 0.32
FBP1 P09467 1/20 0.32
RXRB P28702 6/20 0.31
NR1H4 Q96RI1 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RXRG P48443 3/20 0.31
PDE4B Q07343 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3121517 0.84 NR4A2 (0.40) NR4A2TP53RAB9AKLF5SMN1; SMN2
SCHEMBL3129635 0.82 NR4A2 (0.38) NR4A2TP53RAB9AKLF5SMN1; SMN2
SCHEMBL13689101 0.76 POLB (0.35) POLBIKBKBMEN1KMT2ABMP1
SCHEMBL3742227 0.71 POLB (0.44) POLBIKBKBBMP1FBP1KDM4E
SCHEMBL24158855 0.69 NR4A2 (0.40) NR4A2TP53RAB9AKLF5SMN1; SMN2
SCHEMBL3466896 0.68 POLB (0.34) POLBIKBKBBMP1FBP1KDM4E
SCHEMBL18781937 0.67 HCRTR1 (0.38)
SCHEMBL4664039 0.67 NR4A2 (0.41) NR4A2TP53RAB9AKLF5SMN1; SMN2
SCHEMBL3822091 0.66 NPSR1 (0.31) KDM4EALDH1A1
SCHEMBL13056607 0.66 POLB (0.39) POLBIKBKBBMP1FBP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed