SCHEMBL3133172

SCHEMBL3133172

Cc1cc(Nc2ncc3ncn([C@@H](CO)c4ccc(F)cc4)c3n2)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 6/20 0.46
KCNH2 Q12809 1/20 0.42
JAK2 O60674 9/20 0.42
JAK3 P52333 8/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C8 P10632 3/20 0.42
CYP2C9 P11712 3/20 0.42
JAK1 P23458 3/20 0.42
TYK2 P29597 3/20 0.42
CYP2C19 P33261 3/20 0.42
ADORA3 P0DMS8 2/20 0.42
CYP1A2 P05177 1/20 0.42
PLK4 O00444 5/20 0.39
PAK4 O96013 1/20 0.39
LIMK1 P53667 1/20 0.38
LIMK2 P53671 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3132402 0.87 NTRK1 (0.46) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3132425 0.87 NTRK1 (0.46) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3134973 0.86 NTRK1 (0.55) NTRK1
SCHEMBL3137061 0.85 KCNH2 (0.54) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3137082 0.85 KCNH2 (0.54) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3124459 0.84 NTRK1 (0.51) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3124443 0.84 NTRK1 (0.51) NTRK1KCNH2JAK2JAK3CYP3A4
SCHEMBL3022265 0.76 KCNH2 (0.68) NTRK1KCNH2JAK2JAK3
SCHEMBL3263756 0.74 NTRK1 (0.41) NTRK1KCNH2JAK2JAK3
SCHEMBL28766462 0.74 NTRK1 (0.41) NTRK1KCNH2JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853602-B1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2010-07-14 EP disclosed