SCHEMBL3138762

SCHEMBL3138762

CS(=O)(=O)c1ccc(F)cc1C(=O)N1CCC(CCS(=O)(=O)c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 20/20 0.76
NR1I2 O75469 7/20 0.76
CYP3A4 P08684 3/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035326 0.92 CACNA1B (0.77) CACNA1BNR1I2CYP3A4
SCHEMBL3036818 0.86 CACNA1B (1.00) CACNA1BNR1I2CYP3A4
SCHEMBL3025680 0.84 CACNA1B (0.73) CACNA1BNR1I2CYP3A4
SCHEMBL3128912 0.83 CACNA1B (0.52) CACNA1BNR1I2CYP3A4
SCHEMBL3025687 0.82 CACNA1B (0.73) CACNA1BNR1I2CYP3A4
SCHEMBL3031561 0.81 CACNA1B (0.82) CACNA1BNR1I2CYP3A4
SCHEMBL3032066 0.80 CACNA1B (0.72) CACNA1BNR1I2CYP3A4
SCHEMBL3134634 0.80 CACNA1B (0.65) CACNA1BNR1I2CYP3A4
SCHEMBL3129363 0.80 KMT2A (0.51) CACNA1BNR1I2CYP3A4
SCHEMBL3025559 0.79 CACNA1B (0.86) CACNA1BNR1I2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205083-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO claimed