SCHEMBL31435941

SCHEMBL31435941

CCc1[nH]c2ncc(-c3cn(C4CCN(C)CC4)nc3OC)cc2c1-c1cccc(C(F)F)c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.32
GSK3B P49841 3/20 0.32
CDK9 P50750 3/20 0.32
FGFR1 P11362 2/20 0.32
PLK4 O00444 1/20 0.32
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32
EPHB6 O15197 1/20 0.32
RPS6KA4 O75676 1/20 0.32
STK16 O75716 1/20 0.32
STK10 O94804 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
NTRK1 P04629 1/20 0.32
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
YES1 P07947 1/20 0.32
LYN P07948 1/20 0.32
RET P07949 1/20 0.32
HCK P08631 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31435991 0.84 TLR9 (0.38) AXLGSK3BCHEK1RETFGFR3
SCHEMBL31435981 0.84 MAP4K1 (0.47) MAP3K11MAP4K1IL2
SCHEMBL31435951 0.82 JAK2 (0.39) AXLGSK3BCDK9MAP4K3JAK2
SCHEMBL31435964 0.81 JAK2 (0.39) AXLCDK9MAP4K3JAK2JAK1
SCHEMBL31435948 0.80 JAK2 (0.43) AXLCDK9MAP4K3JAK2JAK1
SCHEMBL31435972 0.79 ELANE (0.32) AXLACVR1GRIN2BGRIN1ELANE
SCHEMBL31435952 0.76 CHEK1 (0.37) AXLGSK3BFGFR1CHEK1RET
SCHEMBL31435943 0.75 KIT (0.52) AXLGSK3BIRAK4MAP4K1IL2
SCHEMBL31435904 0.75 PTPN11 (0.39) AXLACVR1MAP4K1GRIN2BGRIN1
SCHEMBL31435906 0.73 MAP4K1 (0.43) MAP4K1IL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250019378-A1 PYRROLE[2,3-B]PYRIDINE DERIVATIVES AS TYRO3 INHIBITORS HALIA THERAPEUTICS INC (US) 2025-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250019378-A1 PYRROLE[2,3-B]PYRIDINE DERIVATIVES AS TYRO3 INHIBITORS TYRO3, TH, TYR AXL 22/4885GSK3B 342/4885CDK9 2563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.