SCHEMBL3145903

SCHEMBL3145903

CNC1(COc2cnc(C)c(-c3ccc(C#N)cc3)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 12/20 0.44
MAOB P27338 1/20 0.44
AKT1 P31749 1/20 0.44
KCNH2 Q12809 2/20 0.43
RCOR1 Q9UKL0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3780151 0.99 KDM1A (0.44) KDM1AMAOBAKT1KCNH2RCOR1
SCHEMBL3151899 0.91 KDM1A (0.44) KDM1AMAOBAKT1KCNH2RCOR1
Hydrochloric Acid SCHEMBL3843137 0.90 KDM1A (0.44) KDM1AMAOBAKT1KCNH2RCOR1
SCHEMBL3141651 0.89 KDM1A (0.56) KDM1AMAOBAKT1KCNH2RCOR1
SCHEMBL3137179 0.88 CYP1A2 (0.40) KDM1A
SCHEMBL3151443 0.88 KDM1A (0.43) KDM1AMAOBAKT1KCNH2RCOR1
Hydrochloric Acid SCHEMBL3778970 0.88 KDM1A (0.55) KDM1AMAOBAKT1KCNH2RCOR1
Hydrochloric Acid SCHEMBL3776431 0.87 CYP1A2 (0.40) KDM1A
Hydrochloric Acid SCHEMBL3779588 0.87 KDM1A (0.42) KDM1AMAOBAKT1KCNH2RCOR1
Hydrochloric Acid SCHEMBL3778995 0.84 CHRNB4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed