SCHEMBL3166278

SCHEMBL3166278

Nc1nc([AsH]C2CCCN(c3nc(-c4ccc(F)cc4F)cn4ncnc34)C2)ccc1C(=O)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.33
ACKR3 P25106 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
KMT2A Q03164 1/20 0.30
KIT P10721 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4284332 0.85 GSK3B (0.35) PDE2AACKR3ADORA2AADORA1KIT
SCHEMBL8037163 0.73 GSK3B (0.47) KIT
Hydrochloric Acid SCHEMBL4281336 0.73 GSK3B (0.46) KIT
Hydrochloric Acid SCHEMBL4292984 0.71 ADORA2A (0.34) ADORA2AADORA1
SCHEMBL3166285 0.70
SCHEMBL8039872 0.64 GSK3B (0.39)
Hydrochloric Acid SCHEMBL4287764 0.64 GSK3B (0.38)
SCHEMBL2984544 0.61 F2RL3 (0.43) ADORA2AADORA1KMT2A
SCHEMBL2935927 0.59 GSK3B (0.45) KIT
SCHEMBL2246653 0.58 GSK3B (0.34) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229392-A1 TRIAZOLOTRIAZINES AND TRIAZOLOPYRAZINES AND THEIR USE AS GSK3BETA INHIBITORS Bayer Schering Pharma Aktiengesellschaft (DE) 2010-09-22 EP disclosed
WO-2009074259-A1 TRIAZOLOTRIAZINES AND TRIAZOLOPYRAZINES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-06-18 WO disclosed