SCHEMBL3168908

SCHEMBL3168908

Cc1cc(C(C)(C)Sc2cccc(C(=O)O)c2)ccc1OCc1c(C(C)C)nnn1-c1c(Cl)cccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.54
MRGPRX4 Q96LA9 10/20 0.42
PPARA Q07869 1/20 0.35
TYMS P04818 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
MITF O75030 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
KMT2A Q03164 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3168928 0.93 NR1H4 (0.53) NR1H4MRGPRX4
SCHEMBL3164116 0.90 NR1H4 (0.63) NR1H4MRGPRX4
SCHEMBL3164073 0.89 NR1H4 (0.46) NR1H4MRGPRX4MEN1KMT2A
SCHEMBL3159617 0.87 NR1H4 (0.47) NR1H4MRGPRX4PPARA
SCHEMBL3168706 0.85 NR1H4 (0.61) NR1H4MRGPRX4
SCHEMBL3164369 0.82 NR1H4 (0.60) NR1H4
SCHEMBL498196 0.82 NR1H4 (0.48) NR1H4MRGPRX4
SCHEMBL3164122 0.81 NR1H4 (0.57) NR1H4MRGPRX4TYMS
SCHEMBL496925 0.79 NR1H4 (0.53) NR1H4MRGPRX4MEN1KMT2A
SCHEMBL3168921 0.79 NR1H4 (0.55) NR1H4MRGPRX4PPARATYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed