SCHEMBL3172183

SCHEMBL3172183

O=C(O)c1ccccc1S(=O)(=O)c1ccc(C=Cc2ccc(F)cc2F)cc1

nearest known ligand 0.81

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 0.81
HTR2C P28335 10/20 0.81
KCNH2 Q12809 8/20 0.71
NFE2L2 Q16236 4/20 0.50
CYP2D6 P10635 1/20 0.50
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
MMP16 P51512 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3172177 1.00 HTR2A (0.81) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3157651 0.90 HTR2A (1.00) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3157660 0.90 HTR2A (1.00) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3166639 0.90 HTR2A (0.80) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3166649 0.90 HTR2A (0.80) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3162397 0.88 CYP2D6 (0.63) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3162407 0.88 CYP2D6 (0.63) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3152195 0.87 HTR2A (0.75) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3159665 0.87 HTR2A (0.75) HTR2AHTR2CKCNH2NFE2L2CYP2D6
SCHEMBL3151910 0.84 HTR2A (0.72) HTR2AHTR2CKCNH2NFE2L2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807393-B1 DIARYLSULFONES AS 5-HT2A ANTAGONISTS MERCK SHARP & DOHME (GB) 2010-03-31 EP claimed