SCHEMBL31814

SCHEMBL31814

Cc1ccsc1C(=O)Nc1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)ccc1/C=C/c1n[nH]c2ccccc12

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.71
AURKB Q96GD4 4/20 0.71
TBK1 Q9UHD2 11/20 0.38
NSD2 O96028 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
IDO2 Q6ZQW0 1/20 0.38
PCSK9 Q8NBP7 1/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CHEK1 O14757 1/20 0.36
IKBKE Q14164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4317450 0.90 AURKA (0.76) AURKAAURKBTBK1CDK5CDK5R1
SCHEMBL4317456 0.90 AURKA (0.76) AURKAAURKBTBK1CDK5CDK5R1
SCHEMBL4313197 0.89 AURKA (0.74) AURKAAURKBCDK5CDK5R1
SCHEMBL4313205 0.89 AURKA (0.74) AURKAAURKBCDK5CDK5R1
SCHEMBL4313874 0.89 AURKA (0.79) AURKAAURKBCDK5CDK5R1CHEK1
SCHEMBL4316361 0.89 AURKA (0.56) AURKAAURKB
SCHEMBL4322572 0.89 AURKA (0.56) AURKAAURKBTBK1CHEK1IKBKE
SCHEMBL4313866 0.89 AURKA (0.79) AURKAAURKBCDK5CDK5R1CHEK1
SCHEMBL4316358 0.89 AURKA (0.56) AURKAAURKB
Kw-2450 Free Base SCHEMBL4314873 0.89 AURKA (0.87) AURKAAURKBTBK1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012026511-A1 PHARMACEUTICAL COMPOSITION 協和発酵キリン株式会社 (JP) 2012-03-01 WO disclosed