SCHEMBL320163

SCHEMBL320163

CCc1ccc(-c2noc(-c3ccc(-c4ccccc4C(F)(F)F)c(C)c3)n2)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.67
S1PR3 Q99500 3/20 0.51
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16705110 0.91 S1PR1 (0.69) S1PR1S1PR3
SCHEMBL14926465 0.90 S1PR1 (0.74) S1PR1S1PR3NPC1RAB9A
SCHEMBL27904564 0.86 S1PR1 (0.69) S1PR1S1PR3
SCHEMBL319532 0.83 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL557673 0.83 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL10208209 0.83 S1PR1 (0.69) S1PR1S1PR3
Hydrochloric Acid SCHEMBL27904558 0.82 S1PR1 (0.64) S1PR1S1PR3
SCHEMBL13601853 0.82 S1PR1 (0.64) S1PR1S1PR3
SCHEMBL320159 0.82 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL27922398 0.82 S1PR1 (0.67) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590956-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS Merck Serono S.A. (CH) 2013-05-15 EP disclosed
WO-2012004287-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS MERCK SERONO S.A. (CH) 2012-01-12 WO disclosed