SCHEMBL320193

SCHEMBL320193

CC(C)(C)[Si](C)(C)OCC(NCC(=O)O)c1ccc(C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 2/20 0.38
CTSG P08311 2/20 0.38
CTRB1 P17538 2/20 0.38
CMA1 P23946 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EEF2K O00418 1/20 0.37
EGLN1 Q9GZT9 6/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
HTT P42858 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
MMP2 P08253 2/20 0.34
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL319802 0.88 ABCB1 (0.40) EGLN1ADRB2ADRB1ADRB3HTT
SCHEMBL320420 0.84 ABCB1 (0.38) EGLN1ADRB2ADRB1ADRB3HTT
SCHEMBL12505586 0.80 MAN2B1 (0.32)
SCHEMBL320281 0.79 ABCB1 (0.41) ADRB2ADRB1ADRB3HTTCTSL
SCHEMBL321238 0.76 KDM4E (0.47) KDM4EGAAMAPTL3MBTL1EEF2K
SCHEMBL320421 0.74 PRSS1 (0.31) PRSS1CTSGCTRB1CMA1ADRB2
SCHEMBL26648284 0.74 CYP26A1 (0.31)
SCHEMBL26648279 0.74 CYP26A1 (0.31)
SCHEMBL26648513 0.73 ACACB (0.34)
SCHEMBL26648512 0.73 ACACB (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590956-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS Merck Serono S.A. (CH) 2013-05-15 EP disclosed
WO-2012004287-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS MERCK SERONO S.A. (CH) 2012-01-12 WO disclosed