SCHEMBL3203383

SCHEMBL3203383

C1=Cn2c(cc3ccccc32)CN=C1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.37
HTR2A P28223 5/20 0.35
HTR2C P28335 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017480 0.79 NOTUM (0.41) NOTUMHTR2AHTR2C
SCHEMBL1873666 0.69 NOTUM (0.42) NOTUMHTR2AHTR2C
SCHEMBL15466517 0.67 NOTUM (0.43) NOTUMHTR2AHTR2C
SCHEMBL10960778 0.67 NOTUM (0.37) NOTUMHTR2AHTR2C
SCHEMBL10917532 0.66 HTR2A (0.39) NOTUMHTR2AHTR2C
SCHEMBL3050639 0.66 HTR2A (0.44) NOTUMHTR2AHTR2C
SCHEMBL11622046 0.66 NOTUM (0.39) NOTUMHTR2AHTR2C
Hydroxyamine SCHEMBL9656514 0.66 NOTUM (0.39) NOTUMHTR2AHTR2C
SCHEMBL11033039 0.65 HTR2A (0.36) NOTUMHTR2AHTR2C
SCHEMBL4503588 0.64 KMT2A (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790712-B2 Substituted [1,4]diazepino[1,2-A]indoles and azepino[1,2-A]indoles as anti-cytokine inhibitors BOEHRINGER INGELHEIM PHARMACEUTICAL, INC. (US) 2010-09-07 US disclosed