SCHEMBL3204040

SCHEMBL3204040

Cc1ccc(NC(=O)Nc2cc(C(C)(C)C)oc2C(=O)N2CCNC(=O)C2(C)C)cc1-c1ccc(OCCN(C)C)nc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 4/20 0.38
MAPK14 Q16539 4/20 0.37
RAF1 P04049 4/20 0.37
RET P07949 2/20 0.35
KDR P35968 4/20 0.34
KIT P10721 1/20 0.34
FGFR3 P22607 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
CD38 P28907 1/20 0.33
PAICS P22234 1/20 0.33
BRAF P15056 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3210187 0.85 MAPK14 (0.43) FLT3MAPK14RETBRAF
SCHEMBL13487801 0.85 FLT3 (0.34) FLT3RAF1KDRKITFGFR3
SCHEMBL13487767 0.84 RAF1 (0.42) FLT3MAPK14RAF1BRAF
SCHEMBL3212687 0.82 MAPK14 (0.43) MAPK14RETKDRFGFR3BRAF
SCHEMBL3195845 0.77 RAF1 (0.46) MAPK14RAF1
SCHEMBL3200481 0.76 MAPK14 (0.41) FLT3MAPK14RETKDRKIT
SCHEMBL3209489 0.76 MAPK14 (0.47) MAPK14RETKDRFGFR3BRAF
SCHEMBL3218578 0.76 MAPK14 (0.42) FLT3MAPK14
SCHEMBL3208082 0.76 MAPK14 (0.42) FLT3MAPK14KDRKIT
SCHEMBL3198328 0.75 FLT3 (0.41) FLT3MAPK14RETKDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010019930-A1 UREA DERIVATIVES AS INHIBITORS OF MAP KINASES LOCUS PHARMACEUTICALS, INC. (US) 2010-02-18 WO disclosed
US-20100041642-A1 UREA INHIBITORS OF MAP KINASES LOCUS PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed
US-20100041642-A1 UREA INHIBITORS OF MAP KINASES LOCUS PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed
US-20100041642-A1 UREA INHIBITORS OF MAP KINASES LOCUS PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041642-A1 UREA INHIBITORS OF MAP KINASES MAP4K2, MAP3K1, MAP3K20 FLT3 1178/4885MAPK14 33/4885RAF1 74/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.