SCHEMBL3228574

SCHEMBL3228574

Cc1ccc(N(C(=O)CCCCCC(N)=O)c2ccc(C#N)cc2N)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.36
HCRTR2 O43614 1/20 0.36
RORC P51449 5/20 0.33
KDM1A O60341 6/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2A6 P11509 1/20 0.33
PGR P06401 1/20 0.32
AR P10275 1/20 0.31
HDAC3 O15379 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3241012 0.91 ITK (0.36) ITKHCRTR2RORCKDM1AALDH1A1
SCHEMBL3234039 0.87 HDAC3 (0.34) ALDH1A1HDAC3
SCHEMBL3235377 0.83 HDAC3 (0.42) HCRTR2ALDH1A1HDAC3
SCHEMBL3231994 0.81 HDAC3 (0.41) ALDH1A1HDAC3
SCHEMBL3233805 0.80 KDM4E (0.36) ALDH1A1HDAC3
SCHEMBL2122406 0.80 HDAC1 (0.42) ALDH1A1HDAC3
SCHEMBL3235399 0.80 HDAC3 (0.35) ALDH1A1HDAC3
SCHEMBL3237799 0.79 HDAC3 (0.36) HCRTR2ALDH1A1HDAC3
SCHEMBL3232050 0.76 HDAC3 (0.40) HCRTR2ALDH1A1HDAC3
SCHEMBL3068615 0.75 PARP15 (0.38) ITKHCRTR2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed