SCHEMBL3239377

SCHEMBL3239377

CCCC(=O)c1cc(C#N)c(N2CCC(C(=O)OC(C)(C)C)CC2)nc1COCc1ccc(OC)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 17/20 0.48
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2C9 P11712 2/20 0.40
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3229431 0.90 P2RY12 (0.52) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3230375 0.81 P2RY12 (0.62) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3231241 0.79 P2RY12 (0.60) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL4161320 0.78 P2RY12 (0.47) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3234380 0.77 P2RY12 (0.61) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3232013 0.73 SMN1; SMN2 (0.42) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3326980 0.73 P2RY12 (0.72) P2RY12CYP2C9CYP3A4
SCHEMBL4165236 0.73 P2RY12 (0.43) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3229240 0.72 P2RY12 (0.59) P2RY12ALDH1A1KDM4EGAAMAPT
SCHEMBL3223767 0.71 P2RY12 (0.49) P2RY12ALDH1A1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005384-A1 KETONE PYRIDINE ANALOGUES AND THEIR USE IN THE TREATMENT OF CARDIOVASCULAR DISORDERS ASTRAZENECA AB (SE) 2010-01-14 WO disclosed