Doxorubicin

Doxorubicin

SCHEMBL3242

COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(=O)CO)C[C@@H]3O[C@H]1C[C@H](N)[C@H](O)[C@H](C)O1.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP2A

The experimentally established mechanism targets of Doxorubicin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A known ✓ P11388 5/20 1.00
MEN1 O00255 9/20 1.00
KMT2A Q03164 9/20 1.00
THRB P10828 8/20 1.00
BLM P54132 8/20 1.00
RECQL P46063 7/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
HIF1A Q16665 6/20 1.00
TDP1 Q9NUW8 6/20 1.00
BRCA1 P38398 6/20 1.00
MAPT P10636 6/20 1.00
S100A4 P26447 6/20 1.00
MAPK1 P28482 4/20 1.00
USP2 O75604 4/20 1.00
CYP3A4 P08684 4/20 1.00
STAT6 P42226 4/20 1.00
PAX8 Q06710 4/20 1.00
KDM4E B2RXH2 3/20 1.00
ALDH1A1 P00352 3/20 1.00
ABCB1 P08183 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Doxorubicin SCHEMBL317301 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL9335136 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL6251124 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL571906 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL317302 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL6423994 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Doxorubicin SCHEMBL57097 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL21669731 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Epirubicin SCHEMBL21669733 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL
Doxorubicin SCHEMBL5324652 1.00 MEN1 (1.00) MEN1KMT2ATHRBBLMRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 150858 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116983261-B Choline amino acid ionic liquid microemulsion, and preparation method and application thereof NORTHEASTERN UNIVERSITY (CN) 2026-05-26 CN claimed
CN-121846314-B ZIF-8 nano drug delivery system carrying doxorubicin and siTDRKH together and preparation method and application thereof TONGJI HOSPITAL AFFILIATED TO TONGJI MEDICAL COLLEGE OF HUAZHONG UNIVERSITY OF SCIENCE & TECHNOLOGY (CN) 2026-05-26 CN claimed
CN-117050302-B Angiopep-2 modified fluorescent polyamide-amine dendrimer, preparation method thereof and preparation method of nanoparticle based on same XI'AN JIAOTONG UNIVERSITY (CN) 2026-05-26 CN claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
EP-4744665-A1 COMBINATION OF POLQ INHIBITOR COMPOUND AND ANTI-CANCER THERAPEUTIC AGENT OR RADIOTHERAPY Simcere Zaiming Pharmaceutical Co., Ltd. (CN) 2026-05-20 EP claimed
EP-4745155-A1 POWDER CONTAINING PARTICLES OF GELATIN DERIVATIVE AND APPLICATION OF SAME IN MEDICAL TREATMENT National Institute for Materials Science (JP) 2026-05-20 EP claimed
US-12630593-B2 Method of killing leukemia cells by administration of recombinant'Y3 proteins UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2026-05-19 US claimed
CN-117186424-B Hydrogel delivery system based on dextran groups and zwitterionic groups and anti-tumor preparation 山东大学 2026-05-19 CN claimed
US-12629394-B2 Atlas of Choroid Plexus cell types and therapeutic and diagnostic uses thereof THE BROAD INSTITUTE, INC. (US) 2026-05-19 US claimed
CN-116459236-B Controlled release drug implant, preparation method thereof and application thereof in preparation of auxiliary drug for breast cancer postoperative treatment 南京工业大学 2026-05-15 CN claimed
EP-0038357-A4 HYDROLYTIC ENZYME-ACTIVATIBLE PRO-DRUGS. UNIV ILLINOIS (US) 1982-03-22 EP claimed
US-4298594-A BENEFICIAL ALTERATION OF PHARMACODYNAMICS ARTHUR D. LITTLE, INC. (US) 1981-11-03 US claimed
EP-0038357-A1 HYDROLYTIC ENZYME-ACTIVATIBLE PRO-DRUGS University of Illinois Foundation (US) 1981-10-28 EP claimed
US-4267163-A CAUSED BY ADRIAMYCIN CYTOSTATS BIOCARN LIMITED (US) 1981-05-12 US claimed
WO-1981001145-A1 HYDROLYTIC ENZYME-ACTIVATIBLE PRO-DRUGS UNIV ILLINOIS (US) 1981-04-30 WO claimed
US-4263279-A ANTICANCER AGENTS LINKED TO TUMOR-SPECIFIC ANTIBODIES YEDA RESEARCH & DEVELOPMENT CO. LTD (IL) 1981-04-21 US claimed
US-4263428-A LINKING TWO ANTIBIOTICS WITH A DIHYDRAZIDE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1981-04-21 US claimed
EP-0010964-A1 Ravidomycin, process of preparation and pharmaceutical compositions containing same AYERST, MCKENNA AND HARRISON INC. (CA) 1980-05-14 EP claimed
US-4093607-A ANTITUMOR ANTIBODY, ANTICANCER DRUG YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 1978-06-06 US claimed
US-4003996-A Spirolactone for inhibiting the cardiotoxic effects of adriamycin G. D. SEARLE & CO. (US) 1977-01-18 US claimed