SCHEMBL3242007

SCHEMBL3242007

CCCC(NC(=O)O)C(=O)N[C@H]1CC[C@@H]2CN(Cc3ccc(C(F)(F)F)cc3)C[C@@H]21

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 17/20 0.58
KCNH2 Q12809 2/20 0.53
SCN9A Q15858 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2841808 1.00 CACNA1B (0.58) CACNA1BKCNH2SCN9A
SCHEMBL3243073 1.00 CACNA1B (0.58) CACNA1BKCNH2SCN9A
SCHEMBL2847592 0.92 CACNA1B (0.59) CACNA1BKCNH2SCN9A
SCHEMBL3266327 0.92 CACNA1B (0.59) CACNA1BKCNH2SCN9A
SCHEMBL69129 0.91 CACNA1B (0.56) CACNA1BKCNH2SCN9A
SCHEMBL66786 0.91 CACNA1B (0.70) CACNA1BKCNH2SCN9A
SCHEMBL66873 0.91 CACNA1B (0.70) CACNA1BKCNH2SCN9A
SCHEMBL68533 0.89 CACNA1B (0.53) CACNA1BKCNH2SCN9A
SCHEMBL2844911 0.89 CACNA1B (0.53) CACNA1BKCNH2SCN9A
SCHEMBL2844907 0.89 CACNA1B (0.53) CACNA1BKCNH2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010062927-A2 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-06-03 WO claimed
WO-2010062927-A2 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-06-03 WO disclosed