SCHEMBL3247789

SCHEMBL3247789

CC(C[C@H](C)C(=O)N[C@H]1CC[C@@H]2CN(Cc3ccc(F)cc3)C[C@@H]21)N(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 10/20 0.47
KCNH2 Q12809 2/20 0.43
S1PR1 P21453 1/20 0.40
SIGMAR1 Q99720 2/20 0.36
S1PR5 Q9H228 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2419349 0.92 CACNA1B (0.51) CACNA1BKCNH2
SCHEMBL2418610 0.92 CACNA1B (0.51) CACNA1BKCNH2
SCHEMBL3237926 0.92 CACNA1B (0.51) CACNA1BKCNH2
SCHEMBL16497912 0.92 CACNA1B (0.51) CACNA1BKCNH2
SCHEMBL2847786 0.87 CACNA1B (0.51) CACNA1BKCNH2S1PR1SIGMAR1
SCHEMBL68241 0.87 CACNA1B (0.46) CACNA1BKCNH2S1PR1SIGMAR1S1PR5
SCHEMBL68240 0.87 CACNA1B (0.46) CACNA1BKCNH2S1PR1SIGMAR1S1PR5
SCHEMBL2418250 0.87 CACNA1B (0.51) CACNA1BKCNH2
SCHEMBL2849916 0.84 CACNA1B (0.45) CACNA1BKCNH2S1PR1SIGMAR1S1PR5
SCHEMBL2847790 0.84 CACNA1B (0.45) CACNA1BKCNH2S1PR1SIGMAR1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010062927-A2 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-06-03 WO disclosed