SCHEMBL3248124

SCHEMBL3248124

Cc1ccn(-c2ccc(Cl)c(Cl)c2)c(=O)c1-c1ccc2nc(N)ncc2c1

nearest known ligand 0.83

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 18/20 0.83
KIT P10721 17/20 0.83
SRC P12931 17/20 0.83
KDR P35968 8/20 0.74
ABL1 P00519 1/20 0.67
PDGFRA P16234 1/20 0.67
JAK3 P52333 1/20 0.45
MAPK14 Q16539 1/20 0.45
HSP90AB1 P08238 1/20 0.41
EGFR P00533 1/20 0.38
FGFR1 P11362 1/20 0.38
FGFR2 P21802 1/20 0.38
FGFR4 P22455 1/20 0.38
FGFR3 P22607 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258113 0.94 LCK (0.81) LCKKITSRCKDRABL1
SCHEMBL3254179 0.91 LCK (0.85) LCKKITSRCKDRABL1
SCHEMBL3252405 0.91 LCK (1.00) LCKKITSRCKDRABL1
SCHEMBL3249706 0.89 LCK (1.00) LCKKITSRCKDRABL1
SCHEMBL3256148 0.89 LCK (0.88) LCKKITSRCKDRABL1
SCHEMBL3249502 0.88 LCK (0.82) LCKKITSRCKDRABL1
SCHEMBL1345616 0.88 LCK (0.81) LCKKITSRCKDRABL1
SCHEMBL3252054 0.86 LCK (0.81) LCKKITSRCKDRABL1
SCHEMBL3252037 0.85 LCK (0.88) LCKKITSRCKDRABL1
SCHEMBL3257439 0.85 LCK (1.00) LCKKITSRCKDRABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700607-B2 Substituted pyridone compounds and methods of use AMGEN INC. 2010-04-20 US claimed
EP-2079724-B1 SUBSTITUTED PYRIDONE COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2010-05-26 EP disclosed