SCHEMBL3250708

SCHEMBL3250708

COc1ccc(NC(=O)CNS(=O)(=O)c2ccc(OC)c(OC)c2)c(Cc2ccccc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.58
TSHR P16473 1/20 0.51
KMT2A Q03164 3/20 0.47
HTT P42858 3/20 0.47
F2 P00734 2/20 0.45
MEP1B Q16820 1/20 0.44
TMPRSS6 Q8IU80 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3247755 0.92 MAPK1 (0.59) MAPK1TSHRKMT2AHTTF2
SCHEMBL4867744 0.92 MAPK1 (0.63) MAPK1TSHRKMT2AHTTF2
SCHEMBL3254747 0.91 MAPK1 (0.58) MAPK1TSHRKMT2AHTTF2
SCHEMBL3265848 0.90 MAPK1 (0.57) MAPK1TSHRKMT2AHTTF2
SCHEMBL3252225 0.90 MAPK1 (0.61) MAPK1TSHRKMT2AHTTF2
SCHEMBL3256087 0.89 MAPK1 (0.56) MAPK1TSHRKMT2AHTTF2
SCHEMBL4866249 0.89 MAPK1 (0.56) MAPK1TSHRKMT2AHTTF2
SCHEMBL4870830 0.89 MAPK1 (0.55) MAPK1TSHRKMT2AALDH1A1HPGD
SCHEMBL3254680 0.86 MAPK1 (0.59) MAPK1TSHRKMT2AHTTF2
SCHEMBL3253721 0.86 TSHR (0.48) MAPK1TSHRKMT2AMEP1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776347-B1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI AVENTIS (FR) 2010-05-26 EP disclosed
US-7396958-B2 Sulphonamide derivatives, their preparation and their therapeutic application SANOFI AVENTIS (FR) 2008-07-08 US disclosed
US-20070185136-A1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI-AVENTIS (FR) 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185136-A1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION HCRTR2, GIPR, SSTR2 MAPK1 2674/4885TSHR 29/4885KMT2A 1181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.