SCHEMBL3251127

SCHEMBL3251127

CC(C)N1CCC(Oc2cc3cc(C(=O)N4CCN(C=O)CC4)n(C(C)C)c3cc2Br)CC1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 18/20 0.53
CYP2D6 P10635 1/20 0.53
IKBKB O14920 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3250572 0.90 HRH3 (0.55) HRH3CYP2D6IKBKB
SCHEMBL3248817 0.88 HRH3 (0.54) HRH3CYP2D6IKBKB
SCHEMBL3246548 0.86 HRH3 (0.52) HRH3CYP2D6IKBKB
SCHEMBL1552151 0.86 HRH3 (0.55) HRH3CYP2D6IKBKB
SCHEMBL3240758 0.86 HRH3 (0.51) HRH3CYP2D6IKBKB
SCHEMBL3250410 0.86 HRH3 (0.51) HRH3CYP2D6
SCHEMBL3244361 0.86 HRH3 (0.51) HRH3CYP2D6IKBKB
SCHEMBL3248249 0.84 HRH3 (0.50) HRH3CYP2D6
SCHEMBL3241037 0.84 HRH3 (0.50) HRH3CYP2D6
SCHEMBL3252300 0.84 HRH3 (0.51) HRH3CYP2D6IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118089-B1 INDOL-2-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-05-12 EP disclosed