SCHEMBL3258245

SCHEMBL3258245

CCCCCOc1ccc(NC(=O)N(S)C(=O)c2cnoc2C)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.49
THRB P10828 2/20 0.42
THRA P10827 1/20 0.42
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
DHODH Q02127 2/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
GMNN O75496 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTR1A P08908 1/20 0.40
PIM1 P11309 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAOA P21397 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258918 0.84 S1PR1 (0.50) S1PR1THRBTHRARAB9ANPC1
SCHEMBL2865408 0.82 S1PR1 (0.49) S1PR1THRBTHRARAB9ANPC1
SCHEMBL3260301 0.79 S1PR1 (0.49) S1PR1THRBTHRAHTTCYP2C9
SCHEMBL3257407 0.79 S1PR1 (0.50) S1PR1THRBTHRAHTTCYP2C9
SCHEMBL3257536 0.78 S1PR1 (0.49) S1PR1THRBTHRAHTTCYP2C9
SCHEMBL4518245 0.77 S1PR1 (0.50) S1PR1THRBTHRARAB9ANPC1
SCHEMBL3259065 0.76 S1PR1 (0.49) S1PR1THRBTHRARAB9ANPC1
SCHEMBL3258562 0.74 S1PR1 (0.44) S1PR1RAB9ANPC1SMN1; SMN2TP53
SCHEMBL3260070 0.71 S1PR1 (0.47) S1PR1THRBTHRA
SCHEMBL2861336 0.70 S1PR1 (0.52) S1PR1THRBTHRARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747196-B1 SUBSTITUTED ARYL ACYLTHIOUREAS AND RELATED COMPOUNDS; INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS INC (US) 2010-02-10 EP claimed