SCHEMBL3262595

SCHEMBL3262595

COC(=O)c1cc(OC)ccc1Nc1c(-c2ccc3ncn(C)c(=O)c3c2)c(C)nn1-c1ccccc1C

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 20/20 0.65
ADORA3 P0DMS8 1/20 0.65
ADORA2B P29275 2/20 0.53
ADORA2A P29274 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7940136 0.94 ADORA1 (0.74) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL7937178 0.92 ADORA1 (0.60) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL7940009 0.86 ADORA1 (0.71) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1819126 0.83 ADORA1 (0.74) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1815041 0.83 ADORA1 (0.73) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL5010629 0.83 ADORA1 (0.82) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL3311438 0.81 ADORA1 (0.67) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL7937479 0.80 ADORA1 (0.67) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL7943926 0.80 ADORA1 (0.66) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL1815898 0.80 ADORA1 (0.73) ADORA1ADORA3ADORA2BADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020366-A1 AZABICYCLIC SUBSTITUTED 5-AMINOPYRAZOLES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed
WO-2010020366-A1 AZABICYCLIC SUBSTITUTED 5-AMINOPYRAZOLES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed