SCHEMBL3262697

SCHEMBL3262697

CN1CCN(C)[C@H](c2ccc(Nc3cc(N4CCC[C@H](NC(=O)c5cc6ccccc6s5)C4)cn4ccnc34)nc2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.44
CHRNA7 P36544 4/20 0.37
HTR3A P46098 3/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
LCK P06239 1/20 0.36
JAK3 P52333 1/20 0.36
SYK P43405 3/20 0.36
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3262701 1.00 BTK (0.44) BTKCHRNA7HTR3AHTR1ADRD2
SCHEMBL3262293 0.77 EGFR (0.46) BTKHTR1ADRD2HTR2A
SCHEMBL3262289 0.77 EGFR (0.46) BTKHTR1ADRD2HTR2A
SCHEMBL3260836 0.76 SYK (0.42) BTKLCKJAK3SYK
SCHEMBL3260832 0.76 SYK (0.42) BTKLCKJAK3SYK
SCHEMBL2490974 0.72 BTK (0.46) BTK
SCHEMBL2494089 0.72 BTK (0.46) BTK
SCHEMBL2492896 0.72 BTK (0.46) BTK
SCHEMBL9984931 0.69 BTK (0.44) BTKCHRNA7HTR3AHTR1ADRD2
SCHEMBL9984561 0.69 BTK (0.44) BTKCHRNA7HTR3AHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068806-A1 AMIDE DERIVATIVES AS BTK INHIBITORS IN THE TREATMENT OF ALLERGIC, AUTOIMMUNE AND INFLAMMATORY DISORDERS AS WELL AS CANCER CGI PHARMACEUTICALS, INC. (US) 2010-06-17 WO claimed