SCHEMBL3265408

SCHEMBL3265408

COC(=O)c1ccccc1Nc1c(-c2ccc3ncc(=O)n(C)c3c2)c(C)nn1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 17/20 0.57
ADORA2A P29274 1/20 0.57
ADORA2B P29275 1/20 0.57
ADORA3 P0DMS8 1/20 0.47
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7939176 0.92 ADORA1 (0.59) ADORA1ADORA2AADORA2BADORA3
SCHEMBL3263967 0.85 ADORA1 (0.55) ADORA1ADORA2AADORA2BADORA3TDP1
SCHEMBL7937312 0.77 ADORA1 (0.57) ADORA1ADORA2AADORA2BADORA3
SCHEMBL3261148 0.76 ADORA1 (0.49) ADORA1ADORA2AADORA2BADORA3TDP1
SCHEMBL7942415 0.75 ADORA1 (0.60) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1813615 0.75 ADORA1 (0.71) ADORA1ADORA2AADORA2BADORA3TDP1
SCHEMBL3301647 0.74 ADORA1 (0.65) ADORA1ADORA2AADORA2BADORA3
SCHEMBL7938634 0.73 ADORA1 (0.83) ADORA1ADORA2AADORA2BADORA3
SCHEMBL3306840 0.73 ADORA1 (0.54) ADORA1ADORA2AADORA2BADORA3TDP1
SCHEMBL1815646 0.72 ADORA1 (0.56) ADORA1ADORA2AADORA2BADORA3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020366-A1 AZABICYCLIC SUBSTITUTED 5-AMINOPYRAZOLES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed
WO-2010020366-A1 AZABICYCLIC SUBSTITUTED 5-AMINOPYRAZOLES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed